| (11) | Registration Number: | P20191654 (Patent lapsed due to non-payment of renewal fees) | |
| (21) | File number: | P20191654T |
| Expiration Date: | 14.08.2020 |
| (22) | Date of filing the request: | 13.09.2019 |
| (45) | Patent Publication Date and Gazette Number: | 13.12.2019 |
| (54) | English Title: | 3-CYCLOHEXENYL AND CYCLOHEXYL SUBSTITUTED INDOLE AND INDAZOLE COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF |
| (96) | Number of the European patent application: | EP 13829099.4, 14.08.2013 | |
| (97) | Publication data of the European patent application: | EP 2884976, 24.06.2015, 201526, en | |
| (97) | Publication data of the European patent: | EP 2884976, 24.07.2019, 201930, en | |
| (51) | IPC: | A61K 31/416 (2006.01) |
| | | C07D 231/56 (2006.01) |
| | | C07D 471/04 (2006.01) |
| | | C07D 403/06 (2006.01) |
| | | C07D 401/06 (2006.01) |
| | | A61K 31/496 (2006.01) |
| | | A61K 31/5377 (2006.01) |
| | | A61K 31/454 (2006.01) |
| | | A61P 29/00 (2006.01) |
| | | A61P 37/00 (2006.01) |
| | | C07D 209/26 (2006.01) |
| (73) | Holder(s): | | 1. | Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065, US |
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| (72) | Inventor(s): | | 1. | Kenneth Jay Barr, 261 Commonwealth Avenue, No. 7, Boston, MA 02116, US |
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| | | 2. | John Maclean, 431 Washington Street, Unit 4, Brookline, MA 02446, US |
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| | | 3. | Hongjun Zhang, 8 Town House Drive, Newton, MA 02460, US |
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| | | 4. | Richard Thomas Beresis, Apartment 2504, Building 1, 12504 Shimen 2 Road, 200040 Shanghai, CN |
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| | | 5. | Dongshan Zhang, Shanghai Chem Partner Co. Ltd.No. 10 Building 965 Halei Road, Zhangjiang Hi-tech Park Pudong New Area, 201203 Shanghai, CN |
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| | | 6. | Brian Andresen, 33 Avenue Louis Pasteur, Boston, MA 02115, US |
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| | | 7. | Neville Anthony, 52 Lawrence Street, Northborough, MA 01532, US |
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| | | 8. | Blair Lapointe, 33 Avenue Louis Pasteur, Boston, MA 02115, US |
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| | | 9. | Nunzio Sciammetta, 33 Avenue Louis Pasteur, Boston, MA 02115, US |
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| (74) | Representative: | ZMP IP d.o.o.,
Baruna Trenka 7, 10000 Zagreb, HR
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| (30) | Priority Data: | | (31) | PCT/CN2012/080133 | | (32) | 15.08.2012 | | (33) | WO |
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| (86) | PCT Application Number and Date | PCT/US2013054902; 14.08.2013 |
| (87) | PCT Publication Number and Date | WO2014028597; 20.02.2014 |
| (46) | Publication Date of Translation of a European Patent Claims and the Gazette Number: | 13.12.2019 |
| | Annual fee: | 07.11.2019 for the 7th year | |
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| | | NOT IN FORCE | | | Legal Basis | Prestanak važenja patenta zbog neplaćanja održavanja | | | Not in Force Since | 14.08.2020 | |
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