| (11) | Registration Number: | P20192121 (Validated european patent) | |
| (21) | File number: | P20192121T |
| (22) | Date of filing the request: | 27.11.2019 |
| (45) | Patent Publication Date and Gazette Number: | 21.02.2020 |
| (54) | English Title: | PYRIDO-OXAZINONE DERIVATIVES AS TNAP INHIBITORS |
| (96) | Number of the European patent application: | EP 16775006.6, 07.07.2016 | |
| (97) | Publication data of the European patent application: | EP 3319970, 16.05.2018, 201820, en | |
| (97) | Publication data of the European patent: | EP 3319970, 28.08.2019, 201935, en | |
| (51) | IPC: | C07D 498/04 (2006.01) |
| | | A61K 31/4353 (2006.01) |
| | | A61P 19/00 (2006.01) |
| (73) | Holder(s): | | 1. | Daiichi Sankyo Company, Limited, 3-5-1, Nihonbashi Honcho, Chuo-ku, 103-8426 Tokyo, JP |
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| | | | 2. | Sanford Burnham Prebys Medical Discovery Institute, 10901 N. Torrey Pines Rd., La Jolla, CA 92037, US |
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| (72) | Inventor(s): | | 1. | Shojiro Miyazaki, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 2. | Yuko Yamamoto, c/o DAIICHI SANKYO COMPANY LIMITED, 1-2-58 Hiromachi, Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 3. | Keisuke Suzuki, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 4. | Masaharu Inui, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 5. | Masanori Izumi, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 6. | Kaori Soma, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| | | 7. | Anthony Pinkerton, c/o Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA 92037, US |
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| | | 8. | Taeko Shinozaki, c/o Daiichi Sankyo Company Limited, 1-2-58 Hiromachi Shinagawa-ku, 140-8710 Tokyo, JP |
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| (74) | Representative: | Odvjetnica Gorana Grubišić,
Radnička cesta 52, 10000 Zagreb, HR
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| (30) | Priority Data: | | (31) | 201562190145 P | | (32) | 08.07.2015 | | (33) | US |
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| (86) | PCT Application Number and Date | PCT/US2016041345; 07.07.2016 |
| (87) | PCT Publication Number and Date | WO2017007943; 12.01.2017 |
| (46) | Publication Date of Translation of a European Patent Claims and the Gazette Number: | 21.02.2020 |
| | Annual fee: | 17.06.2025 for the 10th year | |
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