| Basic data
|
| (11) | Registration Number: | P20230377 (Validated european patent) | |
| (21) | File number: | P20230377T |
| (22) | Date of filing the request: | 17.04.2023 |
| (54) | English Title: | KRAS G12C INHIBITORS | |
| (51) | IPC: | C07D 401/06 (2006.01) |
| | | C07D 401/14 (2006.01) |
| (73) | Holder(s): | | 1. | Mirati Therapeutics, Inc., 9393 Towne Centre Drive, Suite 200, San Diego, CA 92121, US |
| |
| | | | 2. | Array BioPharma Inc., 3200 Walnut Street, Boulder, CO 80301, US |
| |
| (72) | Inventor(s): | | 1. | Laurence E. Burgess, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 2. | Matthew Arnold Marx, Mirati Therapetutics Inc., 9393 Towne Center Dr., Suite 200, San Diego, CA 92121, US |
| |
| | | 3. | Tony Pisal Tang, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 4. | Mark Joseph Chicarelli, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 5. | Jay Bradford Fell, c/o Array Biopharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 6. | John P. Fischer, c/o Array Biopharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 7. | Adam Cook, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 8. | Christopher Ronald Smith, 3316 Windbreak Court, San Diego, CA 92130, US |
| |
| | | 9. | James F. Blake, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 10. | Martha E. Rodriguez, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 11. | Guy P.A. Vigers, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 12. | Pavel Savechenkov, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 13. | Macedonio J. Mejia, c/o Array BioPharma Inc., 3200 Walnut St., Boulder, CO 80301, US |
| |
| | | 14. | James Gail Christensen, Mirati Therapetutics Inc., 9393 Towne Centre Dr., Suite 200, San Diego, CA 92121, US |
| |
| (74) | Representative: | Vukmir i suradnici odvjetničko društvo d.o.o., Gramača 2L, 10000 Zagreb, HR
|
| | CPZ - CENTAR ZA PATENTE d.o.o., Kutinska 2, 10000 Zagreb, HR
|
| (30) | Priority Data: | | (31) | 201762586775 P | | (32) | 15.11.2017 | | (33) | US |
|
| (86) | PCT Application Number and Date: | PCT/US2018061060; 14.11.2018 |
| (87) | PCT Publication Number and Date: | WO2019099524; 23.05.2019 |
| (96) | Number of the European patent application: | EP 18879484.6, 14.11.2018 | |
| (97) | Publication data of the European patent: | EP 3710439, 15.02.2023, en | |
| (46) | Publication Date of Translation of a European Patent Claims and the Gazette Number: | 23.06.2023, HGIV 13/2023 |
| | Annual fee: | 16.10.2025 for the 8th year | |
|
| | SPC | |
| (21) | Request Number: | S20240024A |
| (22) | Filing Date: | 04.07.2024 |
| (71) | Applicant(s) | | 1. | ARRAY BIOPHARMA INC., 3200 Walnut Street, Boulder, CO 80301, US | | 2. | MIRATI THERAPEUTICS, INC., 9393 Towne Centre Drive, Suite 200, San Diego, CA 92121, US |
|
| (95) | Product Name: | ADAGRASIB ILI NJEGOVA FARMACEUTSKI PRIHVATLJIVA SOL |
| (43) | Request Publication Date: | 19.07.2024 |
| |