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(54) DERIVATI PIPERIDINONA KAO INHIBITORI MDM2 ZA LIJEČENJE RAKA
Osnovni podaci
 
(11)Registarski broj: P20240055  (Upisani europski patent)
(10) HR P20240055 T1
 1. str.Opis
(21) Broj predmeta: P20240055T
(22) Datum podn. zahtjeva: 11.01.2024
(54) Naziv izuma (eng.):PIPERIDINONE DERIVATIVES AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER 
(51) MKP: C07D 211/40 (2006.01)
  C07D 401/04 (2006.01)
  C07D 401/06 (2006.01)
  C07D 407/04 (2006.01)
  C07D 407/06 (2006.01)
  C07D 409/04 (2006.01)
  C07D 413/06 (2006.01)
  C07D 417/06 (2006.01)
  C07D 471/20 (2006.01)
  C07D 279/02 (2006.01)
  C07D 401/12 (2006.01)
  C07D 498/08 (2006.01)
  C07D 498/20 (2006.01)
  A61K 31/4412 (2006.01)
  A61P 35/00 (2006.01)
(73) Nositelj(i):
1.Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320-1799, US
 
(72) Izumitelj(i):
1.Michael David Bartberger, 4471 Ventura Canyon Avenue D-105, Sherman Oaks, CA 91423, US
 
 
2.Joel McIntosh, 540 Fremont Avenue, Pacifica, CA 94044, US
 
 
3.Ana Gonzalez Buenrostro, 1409 Pershing Avenue, San Mateo, CA 94403, US
 
 
4.Hilary Place Beck, 115 Springdale Way, Emerald Hills, CA 94062, US
 
 
5.Xiaoqi Chen, 970 Blair Court, Palo Alto, CA 94303, US
 
 
6.Richard Victor Connors, 935 Crespi Drive, Pacifica, CA 94044, US
 
 
7.Jeffrey Deignan, 500 29th Street, San Francisco, CA 94131, US
 
 
8.Jason A. Duquette, 460 Bayview Avenue, Millbrae, CA 94030, US
 
 
9.John Eksterowicz, 1845 Church Street, San Francisco, CA 94131, US
 
 
10.Benjamin Fisher, 1020 Yates Way Apt. 313, San Mateo, CA 94403, US
 
 
11.Brian Matthew Fox, 124 Swallowtail Court, Brisbane, CA 94005, US
 
 
12.Jiasheng Fu, 221 Pelican Court, Foster City, CA 94404, US
 
 
13.Zice Fu, 788 Santa Maria Lane, Foster City, CA 94404, US
 
 
14.Felix Gonzalez Lopez De Turiso, 10 De Sabla Road Apt. 509, San Mateo, CA 94402, US
 
 
15.Darin James Gustin, 433 Kehoe Avenue, Half Moon, CA 94019, US
 
 
16.Julie Anne Heath, 6 Ivy Drive, Orinda, CA 94563, US
 
 
17.Xin Huang, 16 Abbott Road, Wellesly, MA 02481, US
 
 
18.Michael Johnson, 409 Clipper Street, San Francisco, CA 94114, US
 
 
19.Frank Kayser, 4150, 17th Street, Apt. 25, San Francisco, CA 94114, US
 
 
20.David John Kopecky, 548 Brannan Street 200, San Francisco, CA 94107, US
 
 
21.Sujen Lai, 1439 Floribunda Avenue 15, Burlingame, CA 94010, US
 
 
22.Yihong Li, 821 Taylor Boulevard, Millbrae, CA 94030, US
 
 
23.Zhihong Li, 467 Anita Drive, Millbrae, CA 94030, US
 
 
24.Jiwen Liu, 250 Trysail Court, Foster City, CA 94404, US
 
 
25.Jonathan Dante Low, 18644 Clark Street 5, Tarzana, CA 91356, US
 
 
26.Brian Stuart Lucas, 133 10th Avenue, San Francisco, CA 94118, US
 
 
27.Zhihua Ma, 733 Celestial Lane, Foster City, CA 94404, US
 
 
28.Lawrence R. McGee, 39 Big Sur Way, Pacifica, CA 94044, US
 
 
29.Dustin McMinn, 255 Kent Road, Pacifica, CA 94044, US
 
 
30.Julio Cesar Medina, 1407 Cedar Street, San Carlos, CA 94070, US
 
 
31.Jeffrey Thomas Mihalic, 300 3rd Street 523, San Francisco, CA 94107, US
 
 
32.Steven Howard Olson, 406 Green Hills Drive, Millbrae, CA 94030, US
 
 
33.Yosup Rew, 828 Juno Lane, Foster City, CA 94404, US
 
 
34.Philip Marley Roveto, 500 29th Street, San Francisco, CA 94131, US
 
 
35.Daqing Sun, 804 Cortez Lane, Foster City, CA 94404, US
 
 
36.Xiaodong Wang, 821 Taylor Boulevard, Millbrae, CA 94030, US
 
 
37.Yingcai Wang, 860 Helen Drive, Millbrae, CA 94030, US
 
 
38.Xuelei Yan, 1120 Nimitz Lane, Foster City, CA 94404, US
 
 
39.Ming Yu, 42 Williams Lane, Foster City, CA 94404, US
 
 
40.Jiang Zhu, 747 Coastland Drive, Palo Alto, CA 94303, US
 
 
41.Xianjun Jiao, 2603 All View Way, Belmont, CA 94002, US
 
 
42.Michael William Gribble, 11 Walter Terrace, Abt. One, Somerville, MA 02145, US
 
(74) Opunomoćenik:ZMP IP d.o.o.,
Baruna Trenka 7, 10000 Zagreb, HR
(30) Podaci o pravu prvenstva:
(31) 201161452578 P (32) 14.03.2011 (33) US
 35182710 P  04.06.2010  US
 35232210 P  07.06.2010  US
(62) Broj i dan prvobitne prijave:EP15159363.9; 03.06.2011 
(62) Broj i dan prvobitne prijave:EP11726581.9; 03.06.2011 
(96) Broj europske prijave:EP 18197155.7, 03.06.2011 
(97) Objava europskog patenta:EP 3483143, 18.10.2023, en 
(46) Dan objave prijevoda patentnih zahtjeva europskog patenta i broj HGIV-a:29.03.2024, HGIV 7/2024
 Održavanje:21.05.2025., za godinu 15. 
 

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