| Osnovni podaci
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| (11) | Registarski broj: | P20240055 (Upisani europski patent) | |
| (21) | Broj predmeta: | P20240055T |
| (22) | Datum podn. zahtjeva: | 11.01.2024 |
| (54) | Naziv izuma (eng.): | PIPERIDINONE DERIVATIVES AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER | |
| (51) | MKP: | C07D 211/40 (2006.01) |
| | | C07D 401/04 (2006.01) |
| | | C07D 401/06 (2006.01) |
| | | C07D 407/04 (2006.01) |
| | | C07D 407/06 (2006.01) |
| | | C07D 409/04 (2006.01) |
| | | C07D 413/06 (2006.01) |
| | | C07D 417/06 (2006.01) |
| | | C07D 471/20 (2006.01) |
| | | C07D 279/02 (2006.01) |
| | | C07D 401/12 (2006.01) |
| | | C07D 498/08 (2006.01) |
| | | C07D 498/20 (2006.01) |
| | | A61K 31/4412 (2006.01) |
| | | A61P 35/00 (2006.01) |
| (73) | Nositelj(i): | | 1. | Amgen Inc., One Amgen Center Drive, Thousand Oaks, CA 91320-1799, US |
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| (72) | Izumitelj(i): | | 1. | Michael David Bartberger, 4471 Ventura Canyon Avenue D-105, Sherman Oaks, CA 91423, US |
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| | | 2. | Joel McIntosh, 540 Fremont Avenue, Pacifica, CA 94044, US |
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| | | 3. | Ana Gonzalez Buenrostro, 1409 Pershing Avenue, San Mateo, CA 94403, US |
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| | | 4. | Hilary Place Beck, 115 Springdale Way, Emerald Hills, CA 94062, US |
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| | | 5. | Xiaoqi Chen, 970 Blair Court, Palo Alto, CA 94303, US |
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| | | 6. | Richard Victor Connors, 935 Crespi Drive, Pacifica, CA 94044, US |
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| | | 7. | Jeffrey Deignan, 500 29th Street, San Francisco, CA 94131, US |
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| | | 8. | Jason A. Duquette, 460 Bayview Avenue, Millbrae, CA 94030, US |
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| | | 9. | John Eksterowicz, 1845 Church Street, San Francisco, CA 94131, US |
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| | | 10. | Benjamin Fisher, 1020 Yates Way Apt. 313, San Mateo, CA 94403, US |
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| | | 11. | Brian Matthew Fox, 124 Swallowtail Court, Brisbane, CA 94005, US |
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| | | 12. | Jiasheng Fu, 221 Pelican Court, Foster City, CA 94404, US |
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| | | 13. | Zice Fu, 788 Santa Maria Lane, Foster City, CA 94404, US |
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| | | 14. | Felix Gonzalez Lopez De Turiso, 10 De Sabla Road Apt. 509, San Mateo, CA 94402, US |
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| | | 15. | Darin James Gustin, 433 Kehoe Avenue, Half Moon, CA 94019, US |
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| | | 16. | Julie Anne Heath, 6 Ivy Drive, Orinda, CA 94563, US |
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| | | 17. | Xin Huang, 16 Abbott Road, Wellesly, MA 02481, US |
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| | | 18. | Michael Johnson, 409 Clipper Street, San Francisco, CA 94114, US |
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| | | 19. | Frank Kayser, 4150, 17th Street, Apt. 25, San Francisco, CA 94114, US |
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| | | 20. | David John Kopecky, 548 Brannan Street 200, San Francisco, CA 94107, US |
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| | | 21. | Sujen Lai, 1439 Floribunda Avenue 15, Burlingame, CA 94010, US |
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| | | 22. | Yihong Li, 821 Taylor Boulevard, Millbrae, CA 94030, US |
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| | | 23. | Zhihong Li, 467 Anita Drive, Millbrae, CA 94030, US |
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| | | 24. | Jiwen Liu, 250 Trysail Court, Foster City, CA 94404, US |
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| | | 25. | Jonathan Dante Low, 18644 Clark Street 5, Tarzana, CA 91356, US |
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| | | 26. | Brian Stuart Lucas, 133 10th Avenue, San Francisco, CA 94118, US |
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| | | 27. | Zhihua Ma, 733 Celestial Lane, Foster City, CA 94404, US |
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| | | 28. | Lawrence R. McGee, 39 Big Sur Way, Pacifica, CA 94044, US |
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| | | 29. | Dustin McMinn, 255 Kent Road, Pacifica, CA 94044, US |
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| | | 30. | Julio Cesar Medina, 1407 Cedar Street, San Carlos, CA 94070, US |
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| | | 31. | Jeffrey Thomas Mihalic, 300 3rd Street 523, San Francisco, CA 94107, US |
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| | | 32. | Steven Howard Olson, 406 Green Hills Drive, Millbrae, CA 94030, US |
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| | | 33. | Yosup Rew, 828 Juno Lane, Foster City, CA 94404, US |
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| | | 34. | Philip Marley Roveto, 500 29th Street, San Francisco, CA 94131, US |
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| | | 35. | Daqing Sun, 804 Cortez Lane, Foster City, CA 94404, US |
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| | | 36. | Xiaodong Wang, 821 Taylor Boulevard, Millbrae, CA 94030, US |
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| | | 37. | Yingcai Wang, 860 Helen Drive, Millbrae, CA 94030, US |
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| | | 38. | Xuelei Yan, 1120 Nimitz Lane, Foster City, CA 94404, US |
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| | | 39. | Ming Yu, 42 Williams Lane, Foster City, CA 94404, US |
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| | | 40. | Jiang Zhu, 747 Coastland Drive, Palo Alto, CA 94303, US |
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| | | 41. | Xianjun Jiao, 2603 All View Way, Belmont, CA 94002, US |
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| | | 42. | Michael William Gribble, 11 Walter Terrace, Abt. One, Somerville, MA 02145, US |
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| (74) | Opunomoćenik: | ZMP IP d.o.o., Baruna Trenka 7, 10000 Zagreb, HR
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| (30) | Podaci o pravu prvenstva: | | (31) | 201161452578 P | | (32) | 14.03.2011 | | (33) | US | | | 35182710 P | | | 04.06.2010 | | | US | | | 35232210 P | | | 07.06.2010 | | | US |
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| (62) | Broj i dan prvobitne prijave: | EP15159363.9; 03.06.2011 | |
| (62) | Broj i dan prvobitne prijave: | EP11726581.9; 03.06.2011 | |
| (96) | Broj europske prijave: | EP 18197155.7, 03.06.2011 | |
| (97) | Objava europskog patenta: | EP 3483143, 18.10.2023, en | |
| (46) | Dan objave prijevoda patentnih zahtjeva europskog patenta i broj HGIV-a: | 29.03.2024, HGIV 7/2024 |
| | Održavanje: | 21.05.2025., za godinu 15. | |
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